Wholesale Bulk 99% Pure Tianeptine Acid Powder CAS 66981-73-5 Raw Material for Sale

Product Description:

Tianeptine Acid Powder (CAS 66981-73-5) is a chemical compound that is structurally related to Tianeptine, a well-known antidepressant used in the treatment of major depressive disorder and anxiety. Tianeptine Acid is a derivative of Tianeptine, and its chemical structure includes a functional group that distinguishes it from the parent compound. It is typically produced as a powder and has applications primarily in scientific research and laboratory studies, where its potential pharmacological properties are explored.

Although Tianeptine Acid itself does not have direct therapeutic uses, its relationship to Tianeptine allows researchers to study its mechanisms of action and effects on the central nervous system (CNS). It is thought that Tianeptine and its derivatives work by influencing the balance of certain neurotransmitters in the brain, particularly serotonin, which plays a crucial role in mood regulation.

In addition to its potential use in the pharmaceutical industry, Tianeptine Acid may also have applications in research into neuroprotection, neuroplasticity, and cognitive enhancement. It has been studied for its ability to modulate stress responses and improve neurogenesis in animal models, though its effectiveness and safety in human applications are still under investigation.

Function:

1. Antidepressant Properties: Tianeptine acid, like its salt forms, is recognized for its antidepressant effects. It works through an atypical mechanism, acting as a selective serotonin reuptake enhancer (SSRE). Unlike traditional antidepressants that block serotonin reuptake, tianeptine enhances its reabsorption, which helps balance mood and alleviate symptoms of depression.

2. Modulation of Glutamate Activity: Tianeptine acid also regulates glutamatergic transmission, particularly through AMPA and NMDA receptors. This modulation plays a critical role in reducing stress-related neural damage and improving neuroplasticity, which is often impaired in mood disorders like depression.

3. Neuroprotective Effects: By enhancing neuroplasticity and reducing the damaging effects of stress on neurons, tianeptine acid is associated with neuroprotection. This can help in preserving cognitive functions and mitigating cognitive decline in individuals with depressive disorders.

4. Anxiolytic Properties: Tianeptine acid shows significant anxiolytic (anti-anxiety) effects, reducing symptoms of anxiety by modulating neurotransmitter activity in the brain, particularly in stress-induced or anxiety-prone individuals.

Dosage:

Tianeptine acid (CAS 66981-73-5) is the free acid form of tianeptine, and its dosage can vary depending on its application, particularly in research or preclinical settings. However, tianeptine sodium and tianeptine sulfate are the most commonly studied and prescribed forms, and their dosing guidelines can provide a reference point. Since the bioavailability and pharmacokinetics of tianeptine acid differ from these forms, the dosage for the acid form would need to be adjusted.

General Dosage Considerations:

Tianeptine Sodium: The usual recommended dose for tianeptine sodium is 12.5 mg taken three times per day for the treatment of depression and anxiety.

Tianeptine Sulfate: Due to its slower release and longer half-life, tianeptine sulfate is typically taken at 25-50 mg once or twice per day.
Tianeptine Acid Dosage:

The exact dosage of tianeptine acid (CAS 66981-73-5) is less established in clinical literature due to its less common use compared to the sodium and sulfate forms. If tianeptine acid is being used in research or experimental settings, the dosage is usually determined by the specific goals of the study, focusing on pharmacodynamic and pharmacokinetic parameters. The conversion from tianeptine sodium or sulfate to tianeptine acid is not straightforward because the acid form might have different absorption rates and bioavailability.

Packing and Shipping:

1~25kgs packaging: Aluminium bag inside, Carton box outside.

25kgs packaging: Plastic bag inside, Fiber drum outside

FAQ:

1.What's your MOQ?
Our MOQ is flexible, usually 10 grams~50 grams for a trial order is acceptable.

2. How to deliver the goods?
≤50kg ship by FedEx/UPS, ≥50kg ship by Air, ≥100kg can be shipped by Sea. If you have special request on delivery, please contact us.

3. What is the shelf life for the products?
Most products shelf life 24-36 months.

4. What's your delivery time?
Usually, shipment will be made within 1-3 days against confirmed order.

5. How about the validity of the offer?
Usually, our offer is valid for 2 week. However, validity might vary between different products.